Discovery of potent p38 alpha MAPK inhibitors through a funnel like workflow combining in silico screening and in vitro validation

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Discovery of potent p38 alpha MAPK inhibitors through a funnel like workflow combining in silico screening and in vitro validation

Author: Astolfi, Andrea; Kudolo, Mark; Brea, Jose; Manni, Giorgia; Manfroni, Giuseppe; Palazzotti, Deborah; Sabatini, Stefano; Cecchetti, Federica; Felicetti, Tommaso; Cannalire, Rolando; Massari, Serena; Tabarrini, Oriana; Loza, Maria Isabel; Fallarino, Francesca; Cecchetti, Violetta; Laufer, Stefan A.; Barreca, Maria Letizia
Tübinger Autor(en):
Kudolo, Mark
Laufer, Stefan
Published in: European Journal of Medicinal Chemistry (2019), Bd. 182, Article 111624
Verlagsangabe: Elsevier France - Editions Scientifiques Medicales Elsevier
Language: English
Full text: http://dx.doi.org/10.1016/j.ejmech.2019.111624
ISSN: 1768-3254
DDC Classifikation: 540 - Chemistry and allied sciences
Dokumentart: Article
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